Crystal Structures of ERAP2 Complexed with Inhibitors Reveal Pharmacophore Requirements for Optimizing Inhibitor Potency

Citation:

Mpakali, A. ; Giastas, P. ; Deprez-Poulain, R. ; Papakyriakou, A. ; Koumantou, D. ; Gealageas, R. ; Tsoukalidou, S. ; Vourloumis, D. ; Mavridis, I. M. ; Stratikos, E. ; et al. Crystal Structures Of Erap2 Complexed With Inhibitors Reveal Pharmacophore Requirements For Optimizing Inhibitor Potency. ACS Medicinal Chemistry Letters 2017, 8, 333-337.