Publications by Year: 2010

2010
Agelis, G. ; Roumelioti, P. ; Resvani, A. ; Durdagi, S. ; Androutsou, M. - E. ; Kelaidonis, K. ; Vlahakos, D. ; Mavromoustakos, T. ; Matsoukas, J. An Efficient Synthesis Of A Rationally Designed 1,5 Disubstituted Imidazole At1 Angiotensin Ii Receptor Antagonist: Reorientation Of Imidazole Pharmacophore Groups In Losartan Reserves High Receptor Affinity And Confirms Docking Studies. Journal of Computer-Aided Molecular Design 2010, 24, 749 - 758. Website
Politi, A. P. ; Zervou, M. V. ; Triantafyllidi, H. ; Zoumpoulakis, P. G. ; Mavromoustakos, T. M. ; Zoga, A. A. ; Moutevelis-Minakakis, P. ; Kokotos, G. ; Iliodromitis, E. K. ; Kremastinos, D. T. Hypertension Study In Anaesthetized Rabbits: Protocol Proposal For At 1 Antagonists Screening. JRAAS - Journal of the Renin-Angiotensin-Aldosterone System 2010, 11, 103 - 110. Website
Durdagi, S. ; Papadopoulos, M. G. ; Zoumpoulakis, P. G. ; Koukoulitsa, C. ; Mavromoustakos, T. A Computational Study On Cannabinoid Receptors And Potent Bioactive Cannabinoid Ligands: Homology Modeling, Docking, De Novo Drug Design And Molecular Dynamics Analysis. Molecular Diversity 2010, 14, 257 - 276. Website
Fotakis, C. ; Gega, S. ; Siapi, E. ; Potamitis, C. ; Viras, K. ; Moutevelis-Minakakis, P. ; Kokotos, C. G. ; Durdagi, S. ; Grdadolnik, S. G. ; Sartori, B. ; et al. Interactions At The Bilayer Interface And Receptor Site Induced By The Novel Synthetic Pyrrolidinone Analog Mmk3. Biochimica et Biophysica Acta - Biomembranes 2010, 1798, 422 - 432. Website
Mouchlis, V. D. ; Mavromoustakos, T. M. ; Kokotos, G. Design Of New Secreted Phospholipase A2 Inhibitors Based On Docking Calculations By Modifying The Pharmacophore Segments Of The Fpl67047Xx Inhibitor. Journal of Computer-Aided Molecular Design 2010, 24, 107 - 115. Website
Politi, A. ; Durdagi, S. ; Moutevelis-Minakakis, P. ; Kokotos, G. ; Mavromoustakos, T. Development Of Accurate Binding Affinity Predictions Of Novel Renin Inhibitors Through Molecular Docking Studies. Journal of Molecular Graphics and Modelling 2010, 29, 425 - 435. Website
Mouchlis, V. D. ; Mavromoustakos, T. M. ; Kokotos, G. Molecular Docking And 3D-Qsar Comfa Studies On Indole Inhibitors Of Giia Secreted Phospholipase A2. Journal of Chemical Information and Modeling 2010, 50, 1589 - 1601. Website